Nitrosoureas are organic compounds containing the subunit R2NC(O)N(NO)R, where R can be alkyl, aryl, or H. These compounds are formally derived by the attachment of a nitroso group (NO) to the nitrogen atom of a urea R2NC(O)NR2. Urea is a naturally occurring, innocuous compound, but the nitrosoureas are highly active biochemically. They are sometimes uses for DNA crosslinking.
Examples Examples include:
Arabinopyranosyl-N-methyl-N-nitrosourea (Aranose) Carmustine (BCNU, BiCNU) Chlorozotocin Ethylnitrosourea (ENU) Fotemustine Lomustine (CCNU) Nimustine N-Nitroso-N-methylurea (NMU) Ranimustine (MCNU) Semustine Streptozocin (Streptozotocin) Nitrosourea compounds are DNA alkylating agents and are often used in chemotherapy. They are lipophilic and thus can cross the blood–brain barrier, making them useful in the treatment of brain tumors such as glioblastoma multiforme.
Side effects Some nitrosoureas (e.g. lomustine) have been associated with the development of interstitial lung disease.
References
External links Nitrosourea+Compounds at the U.S. National Library of Medicine Medical Subject Headings (MeSH) Diseases Database (DDB): 9052






