RU-28251, also known as 4,α-methylene-N,N-dipropyltryptamine (4,α-methylene-DPT), is a tricyclic cyclized tryptamine and simplified or partial ergoline. It is a dopamine D2-like receptor agonist and shows affinity for the serotonin 5-HT1 and 5-HT2 receptors (IC50Tooltip half-maximal inhibitory concentration = 141 nM and 723 nM, respectively). The drug inhibits prolactin secretion in animals. The chemical synthesis of RU-28251 has been described. RU-28251 was first described in the scientific literature by 1978.
See also Partial ergoline Bay R 1531 (LY-197206) LY-293284 LY-178210 RU-27849 RU-28306
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