Signaling peptide receptor is a type of receptor which binds one or more signaling peptides or signaling proteins. An example is the tropomyosin receptor kinase B (TrkB), which is bound and activated by the neurotrophic protein brain-derived neurotrophic factor (BDNF). Another example is the μ-opioid receptor (MOR), which is bound and activated by the opioid peptide hormone β-endorphin.
Adiponectin receptor
AdipoR1
Agonists Peptide Adiponectin ADP-355 ADP-399 Non-peptide AdipoRon (–)-Arctigenin Arctiin Gramine Matairesinol Antagonists Peptide ADP-400
AdipoR2
Agonists Peptide Adiponectin ADP-355 ADP-399 Non-peptide AdipoRon Deoxyschizandrin Parthenolide Syringing Taxifoliol Antagonists Peptide ADP-400
Angiotensin receptor
Bradykinin receptor
Agonists Bradykinin Kallidin Antagonists FR-173657 Icatibant LF22-0542
Calcitonin gene-related peptide receptor
Agonists Amylin CGRP Pramlintide Antagonists Atogepant BI 44370 TA CGRP (8-37) MK-3207 Olcegepant Rimegepant SB-268262 Telcagepant Ubrogepant Antibodies Eptinezumab Erenumab Fremanezumab Galcanezumab
Cholecystokinin receptor
CCKA
Agonists Cholecystokinin Antagonists Amiglumide Asperlicin Devazepide Dexloxiglumide Lintitript Lorglumide Loxiglumide Pranazepide Proglumide Tarazepide Tomoglumide
CCKB
Agonists Cholecystokinin CCK-4 Gastrin Pentagastrin (CCK-5) Antagonists Ceclazepide CI-988 (PD-134308) Itriglumide L-365,360 Netazepide Proglumide Spiroglumide
Unsorted Antagonists Nastorazepide
Corticotropin-releasing hormone receptor
CRF1
Agonists Cortagine Corticorelin Corticotropin-releasing hormone Sauvagine Stressin I Urocortin Antagonists Antalarmin Astressin-B CP-154,526 Emicerfont Hypericin LWH-234 NBI-27914 NBI-74788 Pexacerfont R-121919 TS-041 Verucerfont
CRF2
Agonists Corticorelin Corticotropin-releasing hormone Sauvagine Urocortin Antagonists Astressin-B
Cytokine receptor
Endothelin receptor
Agonists Endothelin 1 Endothelin 2 Endothelin 3 IRL-1620 Sarafotoxin Antagonists A-192621 Ambrisentan Aprocitentan Atrasentan Avosentan Bosentan BQ-123 BQ-788 Clazosentan Darusentan Edonentan Enrasentan Fandosentan Feloprentan Macitentan Nebentan Sitaxentan Sparsentan Tezosentan Zibotentan
Galanin receptor
GAL1
Agonists Galanin Galanin (1-15) Galanin-like peptide Galmic Galnon NAX 810-2 Antagonists C7 Dithiepine-1,1,4,4-tetroxide Galantide (M15) M32 M35 M40 SCH-202596
GAL2
Agonists Galanin Galanin (1-15) Galanin (2-11) Galanin-like peptide Galmic Galnon J18 NAX 810-2 Antagonists C7 Galantide (M15) M32 M35 M40 M871
GAL3
Agonists Galanin Galanin (1-15) Galmic Galnon Antagonists C7 Galantide (M15) GalR3ant HT-2157 M32 M35 M40 SNAP-37889 SNAP-398299
Growth hormone secretagogue receptor
Growth hormone receptor
Growth-hormone-releasing hormone receptor
Glucagon-like peptide receptor
GLP-1
Agonists Albiglutide Beinaglutide Dulaglutide Efpeglenatide Exenatide GLP-1 Langlenatide Liraglutide Lixisenatide Oxyntomodulin Pegapamodutide Semaglutide Taspoglutide
GLP-2
Agonists Apraglutide Elsiglutide Glepaglutide GLP-2 Teduglutide
Others Propeptides Preproglucagon Proglucagon
Glucagon receptor
Agonists Dasiglucagon Glucagon Oxyntomodulin Antagonists Adomeglivant L-168,049 LGD-6972 Propeptides Preproglucagon Proglucagon
Gonadotropin-releasing hormone receptor
Gonadotropin receptor
Growth factor receptor
Insulin receptor
Agonists Chaetochromin (4548-G05) Insulin-like growth factor 1 Insulin-like growth factor 2 Insulin Insulin aspart Insulin degludec Insulin detemir Insulin glargine Insulin glulisine Insulin lispro Mecasermin Mecasermin rinfabate Antagonists BMS-754807 S661 S961 Kinase inhibitors Linsitinib Antibodies Xentuzumab (against IGF-1 and IGF-2)
KiSS1-derived peptide receptor
Agonists Kisspeptin (kisspeptin-54, metastin) Kisspeptin-10 KISS1-305 MVT-602 (RVT-602, TAK-448) TAK-683 Antagonists Kisspeptin-234
Leptin receptor
Agonists Leptin Metreleptin
Melanin-concentrating hormone receptor
MCH1
Agonists Melanin-concentrating hormone Antagonists ATC-0065 ATC-0175 GW-803430 NGD-4715 SNAP-7941 SNAP-94847
MCH2
Agonists Melanin-concentrating hormone
Melanocortin receptor
Neuropeptide FF receptor
Agonists Neuropeptide AF Neuropeptide FF Neuropeptide SF (RFRP-1) Neuropeptide VF (RFRP-3) Antagonists BIBP-3226 RF9
Neuropeptide S receptor
Agonists Neuropeptide S Antagonists ML-154 SHA-68
Neuropeptide Y receptor
Y1
Agonists Neuropeptide Y Peptide YY Antagonists BIBO-3304 BIBP-3226 BVD-10 GR-231118 PD-160170
Y2
Agonists 2-Thiouridine 5'-triphosphate Neuropeptide Y Neuropeptide Y (13-36) Peptide YY Peptide YY (3-36) Antagonists BIIE-0246 JNJ-5207787 SF-11
Y4 Agonists GR-231118 Neuropeptide Y Pancreatic polypeptide Peptide YY Antagonists UR-AK49
Y5
Agonists BWX-46 Neuropeptide Y Peptide YY Antagonists CGP-71683 FMS-586 L-152,804 Lu AA-33810 MK-0557 NTNCB Velneperit (S-2367)
Neurotensin receptor
NTS1
Agonists Neurotensin Neuromedin N Antagonists Meclinertant SR-142948
NTS2
Agonists Neurotensin Antagonists Levocabastine SR-142948
Opioid receptor
Orexin receptor
Oxytocin receptor
Prolactin receptor
Parathyroid hormone receptor
Agonists Abaloparatide Parathyroid hormone Parathyroid hormone-related protein (PTHrP) Semparatide Teriparatide
Relaxin receptor
Agonists Insulin-like factor 3 Relaxin (1, 2, 3) Serelaxin
Somatostatin receptor
Tachykinin receptor
Thyrotropin-releasing hormone receptor
Agonists Azetirelin JTP-2942 Montirelin Orotirelin Posatirelin Protirelin Rovatirelin RX-77368 (thymoliberin) Taltirelin TRH (TRF)
Thyrotropin receptor
Agonists Thyrotropin alfa TSH (thyrotropin)
Vasopressin receptor
Vasoactive intestinal peptide receptor and Pituitary adenylate cyclase-activating peptide
VIPR1
Agonists Peptide Bay 55-9837 LBT-3393 PACAP VIP
VIPR2
Agonists Peptide LBT-3627 PACAP VIP
PAC1
Agonists PACAP PACAP (1-27) PACAP (1-38) Antagonists PACAP (6-38)
Unsorted PHI PHM PHV
Others Endogenous Adrenomedullin Apelin Asprosin Bombesin Calcitonin Carnosine CART CLIP DSIP Enteroglucagon Formyl peptide GALP GIP GRP Integrin ligands collagens fibrinogen fibronectin laminins ICAM-1 ICAM-2 osteopontin VCAM-1 vitronectin Kininogens Motilin Natriuretic peptides ANP BNP CNP urodilatin Nesfatin-1 Neuromedin B Neuromedin N Neuromedin S Neuromedin U Obestatin Osteocalcin Resistin Secretin Thymopoietin Thymosins Thymulin Urotensin-II VGF Exogenous Lifitegrast (LFA-1 antagonist)
See also Neuropeptide receptor Neurotransmitter receptor
References
External links Peptide+receptor at the U.S. National Library of Medicine Medical Subject Headings (MeSH)
